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M149

Methiothepin mesylate salt

Name: Methiothepin mesylate salt
Brand: SIGMA

≥98% (HPLC), solid

동의어(들):

1-[10,11-Dihydro-8-(methylthio)dibenzo[b,f]thiepin-10-yl]-4-methylpiperazine mesylate salt, Metitepine mesylate salt

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제품정보 (DICE 배송 시 비용 별도)

Linear Formula:

C₂₀H₂₄N₂S₂ · CH₃SO₃H

CAS 번호:

74611-28-2

Molecular Weight:

452.65

NACRES:

NA.77

PubChem Substance ID:

24278104

UNSPSC Code:

12352200

MDL number:

MFCD00153831

Assay:

≥98% (HPLC)

Form:

solid

Quality level:

100

Storage condition:

desiccated

기술 서비스

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도움 문의

속성

Quality Level

100

assay

≥98% (HPLC)

form

solid

storage condition

desiccated

color

white

solubility

H₂O: 13 mg/mL

SMILES string

CS(O)(=O)=O.CSc1ccc2Sc3ccccc3CC(N4CCN(C)CC4)c2c1

InChI

1S/C20H24N2S2.CH4O3S/c1-21-9-11-22(12-10-21)18-13-15-5-3-4-6-19(15)24-20-8-7-16(23-2)14-17(18)20;1-5(2,3)4/h3-8,14,18H,9-13H2,1-2H3;1H3,(H,2,3,4)

InChI key

CZMDZGZYKOGLJY-UHFFFAOYSA-N

Gene Information

human ... HTR1A(3350), HTR1B(3351), HTR1D(3352), HTR1E(3354), HTR1F(3355), HTR6(3362), HTR7(3363)

설명

General description

Methiothepin belongs to a new class of dibenzothiophenes. Methiothepin possesses neuroleptic activity.

Application

Methiothepin mesylate salt has been used to explore the relationship between circulating cells and the niche. It has also been used in serotonin (5-HT) and antagonists in vivo bioassays and in in vivo antagonist and lipopolysaccharide stimulations.

Biochem/physiol Actions

Methiothepin mesylate salt is a 5-HT₁, 5-HT₆, 5-HT₇ serotonin receptor antagonist, which blocks serotonin autoreceptors.

저장 등급

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

Eyeshields, Gloves, type N95 (US)

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국제 무역 품목 번호

SKU	GTIN
MABN1773	04055977181630
M149-100MG	04061834040682
M149-250MG	04061834040699