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P9233

Piribedil maleate salt

Synonym(s):

2-[4-(1,3-Benzodioxol-5-ylmethyl)-1-piperazinyl]pyrimidine maleate salt

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About This Item

Empirical Formula (Hill Notation):
C20H22N4O6
CAS Number:
937719-94-3
Molecular Weight:
414.41
NACRES:
NA.77
PubChem Substance ID:
24278661
UNSPSC Code:
12352200
MDL number:
MFCD02684412
Form:
powder
Quality level:
100
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form

powder

Quality Level

100

solubility

DMSO: >10 mg/mL, H2O: >10 mg/mL

originator

Servier

storage temp.

2-8°C

SMILES string

[H]\C(=C(/[H])C(O)=O)C(O)=O.C1Oc2ccc(CN3CCN(CC3)c4ncccn4)cc2O1

InChI

1S/C16H18N4O2.C4H4O4/c1-4-17-16(18-5-1)20-8-6-19(7-9-20)11-13-2-3-14-15(10-13)22-12-21-14;5-3(6)1-2-4(7)8/h1-5,10H,6-9,11-12H2;1-2H,(H,5,6)(H,7,8)/b;2-1-

InChI key

DKGOFBARSQSLOW-BTJKTKAUSA-N

Gene Information

human ... DRD3(1814)

Biochem/physiol Actions

A direct dopamine agonist; may be selective for the D3 subtype; no significant affinity for D1 receptors.

Features and Benefits

This compound was developed by Servier. To browse the list of other pharma-developed compounds and Approved Drugs/Drug Candidates, click here.

pictograms

Exclamation mark
GHS07

signalword

Warning

Hazard Classifications

Eye Irrit. 2 - Skin Irrit. 2 - STOT SE 3

target_organs

Respiratory system

Storage Class

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

dust mask type N95 (US), Eyeshields, Gloves

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Certificates of Analysis (COA)

Lot/Batch Number
020K4605

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A Cagnotto et al.
European journal of pharmacology, 313(1-2), 63-67 (1996-10-10)
Receptor binding autoradiography, using the selective ligand [3H]7-OH-(R)DPAT (R(+)-2-dipropylamino-7-hydroxy 1,2,3,4-tetrahydronaphthalene), showed that piribedil is a potent inhibitor at dopamine D3 receptors in limbic regions (island of Calleja), with affinity (IC50) between 30 and 60 nM. The in vitro IC50 of

Global Trade Item Number

SKUGTIN
P9233-10MG04061832083735
P9233-50MG04061832083742